Considering the fact that the fluorine-/boron-containing compounds are omnipresent in medicinal chemistry, hence, research in the Beyondlxw Group merges the powerful synthetic methodologies with recourse to the modern catalysis and medicinal chemistry. Motivation for our work arises from the fundamental interest in elemento-medicinal chemistry, and much emphasis lies with the elucidation of their intrinsic structure and activity relationship, thus exploring the potential drug lead.